Arylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties

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dc.citation.epage450
dc.citation.issue4
dc.citation.journalTitleChemistry & Chemical Technology
dc.citation.spage447
dc.citation.volume12
dc.contributor.affiliationTernopil V. Hnatyuk National Pedagogical University
dc.contributor.affiliationI. Ya. Horbachevsky Ternopil State Medical University
dc.contributor.authorBaranovskyi, Vitaliy
dc.contributor.authorSymchak, Ruslan
dc.contributor.authorPokryshko, Olena
dc.contributor.authorKlymnyuk, Sergiy
dc.contributor.authorGrishchuk, Bogdan
dc.coverage.placenameLviv
dc.date.accessioned2019-06-21T07:58:04Z
dc.date.available2019-06-21T07:58:04Z
dc.date.created2018-01-20
dc.date.issued2018-01-20
dc.description.abstractКупрокаталітичним аніонарилюванням амідів акрилової і метакрилової кислот солями 4-ацетилфе- нілдіазонію синтезовані 3-(4-ацетилфеніл)-(2-метил)-2-хлоро (бромо, тіоціанато)пропанаміди. Циклізацією тіоціанато- амідів одержані арилзаміщені 2-амінотіазол-4(5Н)-они з ацетофеноновим фрагментом. Досліджено протибакте- ріальну та протигрибкову активність синтезованих сполук.
dc.description.abstract13-(4-Acetylphenyl)-(2-methyl)-2-chloro(bromo, thiocyanato)propanamides have been obtained via copper catalytic anionarylation of acrylic and methacrylic acids amides by 4-acetylphenyldiazonium salts. 5-(4-Acetylphenyl) substituted 2-aminothiazol-4(5H)-ones were synthesized by cyclisation of thiocyanatoamides. All synthesized compounds were tested for their antibacterial and antomycotic activity.
dc.format.extent447-450
dc.format.pages4
dc.identifier.citationArylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties / Vitaliy Baranovskyi, Ruslan Symchak, Olena Pokryshko, Sergiy Klymnyuk, Bogdan Grishchuk // Chemistry & Chemical Technology. — Lviv : Lviv Politechnic Publishing House, 2018. — Vol 12. — No 4. — P. 447–450.
dc.identifier.citationenArylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties / Vitaliy Baranovskyi, Ruslan Symchak, Olena Pokryshko, Sergiy Klymnyuk, Bogdan Grishchuk // Chemistry & Chemical Technology. — Lviv : Lviv Politechnic Publishing House, 2018. — Vol 12. — No 4. — P. 447–450.
dc.identifier.urihttps://ena.lpnu.ua/handle/ntb/45209
dc.language.isoen
dc.publisherLviv Politechnic Publishing House
dc.relation.ispartofChemistry & Chemical Technology, 4 (12), 2018
dc.relation.references[1] O'Neil M. (Ed.): The Merck Index: An Encyclopedia of Chemicals, Drugs, and Biologicals, 15th edn. Merck and Co. Inc., Cambridge 2013.
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dc.relation.references[7] Baranovskii V., Simchak R., Grishchuk B.: Russ. J. Gen. Chem.,2009, 79, 269. https://doi.org/10.1134/S1070363209020170
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dc.relation.referencesen[1] O'Neil M. (Ed.): The Merck Index: An Encyclopedia of Chemicals, Drugs, and Biologicals, 15th edn. Merck and Co. Inc., Cambridge 2013.
dc.relation.referencesen[2] Cripps R., Biochem J., 1975, 152, 233.https://doi.org/10.1042/bj1520233
dc.relation.referencesen[3] Salas P., Soto A., Carretero A. et al.:Molecules, 2010, 15,8813. https://doi.org/10.3390/molecules15128813
dc.relation.referencesen[4] Pharmaceutical Manufacturing Encyclopedia. William Andrew Publishing, Norwich, NY 2007.
dc.relation.referencesen[5] Shen Y., Li B., Xu H. et al., Pharmazie, 2013, 68, 307.
dc.relation.referencesen[6] Wang Z., Li X., Xu W. et al.:Med. Chem. Commun., 2015, 6,2146. https://doi.org/10.1039/P.5MD00357A
dc.relation.referencesen[7] Baranovskii V., Simchak R., Grishchuk B., Russ. J. Gen. Chem.,2009, 79, 269. https://doi.org/10.1134/S1070363209020170
dc.relation.referencesen[8] Baranovskii V., Yatsyuk V., Grishchuk B., Russ. J. Gen. Chem.,2014, 84, 1505. https://doi.org/10.1134/S1070363214080106
dc.relation.referencesen[9] Grishchuk B., Baranovskii V., Klymnyuk S. et al., Pharm. Chem. J., 2011, 45, 532. https://doi.org/10.1007/s11094-011-0673-0
dc.relation.referencesen[10] Grishchuk B., Simchak R., Baranovskii V. et al., Pharm. Chem. J., 2013, 47, 307. https://doi.org/10.1007/s11094-013-0949-7
dc.relation.referencesen[11] Grishchuk B., Yatsyuk V., Baranovskii V. et al., Pharm. Chem. J., 2016, 50, 534. https://doi.org/10.1007/s11094-016-1484-0
dc.relation.referencesen[12] Yatsyuk V., Pokryshko O., Yaniv Z. et al., Chem. Chem. Technol., 2015, 9, 193. https://doi.org/10.23939/chcht09.02.193
dc.relation.referencesen[13] Grishchuk B., Baranovskyi V., Klymnyuk S., Pharmac. Rev.,2011, 4, 117.
dc.relation.urihttps://doi.org/10.1042/bj1520233
dc.relation.urihttps://doi.org/10.3390/molecules15128813
dc.relation.urihttps://doi.org/10.1039/C5MD00357A
dc.relation.urihttps://doi.org/10.1134/S1070363209020170
dc.relation.urihttps://doi.org/10.1134/S1070363214080106
dc.relation.urihttps://doi.org/10.1007/s11094-011-0673-0
dc.relation.urihttps://doi.org/10.1007/s11094-013-0949-7
dc.relation.urihttps://doi.org/10.1007/s11094-016-1484-0
dc.relation.urihttps://doi.org/10.23939/chcht09.02.193
dc.rights.holder© Національний університет „Львівська політехніка“, 2018
dc.rights.holder©Baranovskyi V., Symchak R., Pokryshko O., Klymnyuk S.,Grishchuk B., 2018
dc.subjectаніонарилювання
dc.subjectаміди акрилової і метакрилової кислот
dc.subjectсолі 4-ацетилфенілдіазонію
dc.subject5-арилза- міщені 2-амінотіазол-4(5Н)-они
dc.subjectпротимікробна активність
dc.subjectanionarylation
dc.subjectacrylic and methacrylic acids amides
dc.subject4-acetylphenyldiazonium salts
dc.subject5-arylsubstituted 2-aminothiazol-4(5H)-ones
dc.subjectantimicrobial activity
dc.titleArylsubstituted halogen(thiocyanato)amides containing 4-acetylphenyl fragment. Synthesis, cyclization and antimicrobial properties
dc.title.alternativeАрилзаміщені галогено(тіоціанато)аміди, що містять 4-ацетилфенільний фрагмент. Синтез, циклізація та протимікробні властивості
dc.typeArticle

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Chemistry & Chemical Technology. – 2018. – Vol. 12, No. 4